Antazoline
Also known as: Imidamine HCl, Phenazolinum
Antazoline is an ethylendiamine derivative and used as an antihistaminic agent to relieve symptoms and to treat allergic manisfastations. Administered orally.
Primary Characteristics
Antazoline is also known as Imidamine HCl, Phenazolinum.
It is of Synthetic origin and belongs to Imidazole.
It is classified in Anti Allergic Agent pharmacological group. It is also classified under Opthalmic Products .
Molecular Weight: 265.35 · Solubility in Water: sparingly soluble · Solubility in Alcohol: soluble · Non-proprietary name: Antazoline · pH: 4 · Isotonic value: 6.05.

Pharmacokinetics
None recorded.
Advertisement
Indications
Antazoline is primarily indicated in conditions like Allergic conjunctivitis, Insect bites, Skin irritations.
Contraindications
Antazoline is contraindicated in conditions like Heart disease, Narrow-angle glaucoma.
Dosage
Antazoline's dosage details are as follows:
| Dose | Single Dose | Frequency | Route | Instructions |
|---|---|---|---|---|
| Adult Dosage | ||||
| 0.375 mg | 0.375 mg | Every 6h | Ophthalmic | |
| Paediatric Dosage (20kg) | ||||
| 0.375 mg | 0.375 mg | Every 6h | Opthalmic | - |
| Neonatal Dosage (3kg) | ||||
| 0 – 0 | — | — | Not usd in this age group | |
Drug Interactions
Always consult your physician for the change of dose regimen or an alternative drug of choice that may strictly be required.
Side Effects
Antazoline is known to cause more or less tolerable side effects which are usually transient. These include Hypersensitivity reactions.
Warnings / Precautions
Available Brands
Storage Conditions
Drug Classification
- 1.3 — Anti-allergics (Antihistamines) and drugs used in anaphylaxis
- 2.21.6 — Non-specific anticonjunctivitis preparations
- 3.25.4 — Nasal preparations