DrugInfoSys

Brimonidine (Tartrate)

Drug #1615

Brimonidine (Tartrate) is an alpha-2 adrenoceptor stimulant. Brimonidine (Tartrate) is used topically to lower the intra-ocular pressure (IOP) in open angle glaucoma or ocular hypertension in patients for whom beta-blockers are inappropriate or may be given as an adjunct to beta-blocker.

Primary Characteristics

It is of Synthetic origin.

Molecular Weight: 442.2 · Non-proprietary name: Brimonidine (Tartrate) · pH: 6.3.

Molecular structure of Brimonidine (Tartrate)

Pharmacokinetics

None recorded.

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Indications

Brimonidine (Tartrate) is primarily indicated in conditions like Ocular hypertension, Open-angle glaucoma.

Contraindications

Brimonidine (Tartrate) is contraindicated in conditions like Hypersensitivity to the drug.

Dosage

Brimonidine (Tartrate)'s dosage details are as follows:

DoseSingle DoseFrequencyRouteInstructions
Adult Dosage
1 drop1 dropEvery 8hOpthalmicFor open angle galucoma/Occular hypertension
Paediatric Dosage (20kg)
No data.
Neonatal Dosage (3kg)
No data.

Drug Interactions

Unknown3 interactions

Always consult your physician for the change of dose regimen or an alternative drug of choice that may strictly be required.

Side Effects

Brimonidine (Tartrate) is known to cause more or less tolerable side effects which are usually transient. These include Asthenia , Blurred vision, Conjunctival bleeding, Dry mouth, Headache, Hyperemia, Increased tearing, Lid retraction, Lids edema, Mydriasis, Ocular irritation, Taste disturbance.

Warnings / Precautions

It should be used with caution in patients with depression, cerebral or coronary insufficiency, raynauds phenomenon, orthostatic hypotension, severe cardiovascular disease and hepatic or renal impairment. Donot use in patients receiving mono amino oxidase inhbitors.

Available Brands

Click on a strength to view available brands.

Single Ingredient

Multi-Ingredient Combinations

Eye Drops

Storage Conditions

Brimonidine (Tartrate) should be stored Drops.

Drug Classification

  1. 1.21.4.2Beta blockers

Manufacturers

Manufacturers of Brimonidine (Tartrate) in Pakistan: