Fludiazepam
Fludiazepam used for the short-term treatment of anxiety disorders.
Primary Characteristics
It is of Synthetic origin and belongs to Benzodiazapene.
Molecular Weight: 302.7 · pKa: 2.22 · Solubility in Water: slightly soluble · Solubility in Alcohol: soluble · Non-proprietary name: Fludiazepam.

Pharmacokinetics
Absorption: Fludiazepam has an pre-systemic (first-pass) metabolism accounts for 90%.
Elimination: it is metabolised via hepatic, plasma half-life is 10-30 hr, renal excretion is major 24 ± 3.1.
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Indications
Fludiazepam is primarily indicated in conditions like Anxiety.
Contraindications
Fludiazepam is contraindicated in conditions like Hypersensitivity to any component of product.
Dosage
Fludiazepam's dosage details are as follows:
| Dose | Single Dose | Frequency | Route | Instructions |
|---|---|---|---|---|
| Adult Dosage | ||||
| 22.5 mg | 22.5 mg | Every 24h | PO | At bed time. |
| Paediatric Dosage (20kg) | ||||
| No data. | ||||
| Neonatal Dosage (3kg) | ||||
| No data. | ||||
Drug Interactions
None recorded.
Side Effects
The signs and symptoms that are produced after acute overdosage of Fludiazepam are Nausea, Liver damage, Drowsiness, Drowsiness, Hyperglycemia, Hypoglycemia, Dizziness, Coma and death, Abdominal pain, CNS depression, Cerebral edema, Weakness .
Fludiazepam is known to cause more or less tolerable side effects which are usually transient. These include Drowsiness, Headache, Sedation , Slurred speech, Weakness.
Warnings / Precautions
Available Brands
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Single Ingredient
Storage Conditions
Drug Classification
- 1.24.3 — Drugs used in anxiety and sleep disorders
Manufacturers
Manufacturers of Fludiazepam in Pakistan: